CX157

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CX157
CX157 structure.svg
Systematic (IUPAC) name
3-fluoro-7-(2,2,2-trifluoroethoxy)phenoxathiine 10,10-dioxide
Clinical data
Legal status
  • Uncontrolled
Routes of
administration
Oral
Identifiers
ATC code none
PubChem CID: 18687754
ChemSpider 13701383 YesY
Chemical data
Formula C14H8F4O4S
Molecular mass 348.27 g/mol
  • FC(F)(F)COc2cc3Oc1cc(F)ccc1S(=O)(=O)c3cc2
  • InChI=1S/C14H8F4O4S/c15-8-1-3-12-10(5-8)22-11-6-9(21-7-14(16,17)18)2-4-13(11)23(12,19)20/h1-6H,7H2 YesY
  • Key:PDIMOTRDGUQMNY-UHFFFAOYSA-N YesY
  (verify)

CX157 (proposed trade name TriRima, formerly Tyrima) is a selective and reversible inhibitor of MAO-A (RIMA).[1] As of 2007 it was in phase II clinical trials for the treatment of depression.[2] In 2013, it was discontinued for both depression and anxiety.[1]

References

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  2. Clinical trial number NCT00739908 at ClinicalTrials.gov


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