N-Phenethyl-14-ethoxymetopon

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N-Phenethyl-14-ethoxymetopon
N-Phenethyl-14-ethoxymetopon2DCSD.svg
Systematic (IUPAC) name
(5α)-14-Ethoxy-3-hydroxy-5-methyl-17-(2-phenylethyl)-4,5-epoxymorphinan-6-one
Identifiers
PubChem CID: 11049533
Chemical data
Formula C27H31NO4
Molecular mass 433.538 g/mol
  • O=C1CCC2(C3CC4=C(C25CCN3CCC6=CC=CC=C6)C(OC15C)=C(O)C=C4)OCC
  (verify)

N-Phenethyl-14-ethoxymetopon is a drug that is a derivative of metopon. It is a potent analgesic, around 60 times stronger than morphine and produces significantly less constipation.[1]

N-Phenethyl-14-ethoxymetopon acts as an agonist at both μ- and δ-opioid receptors, with a Ki of 0.16nM at μ and 3.14nM at δ.[2]

See also

References

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  2. ↑ Lua error in package.lua at line 80: module 'strict' not found.
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