L-759,656
From Infogalactic: the planetary knowledge core
Systematic (IUPAC) name | |
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(6aR,10aR)-1-methoxy-6,6-dimethyl-9-methylidene-3-(2-methyloctan-2-yl)-7,8,10,10a-tetrahydro-6aH-benzo[c]chromene
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Identifiers | |
PubChem | CID: 5311216 |
IUPHAR/BPS | 749 |
ChemSpider | 4470735 |
ChEMBL | CHEMBL294013 |
Chemical data | |
Formula | C26H40O2 |
Molecular mass | 384.593 g/mol |
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L-759,656 is an analgesic drug that is a cannabinoid agonist. It is a highly selective agonist for the CB2 receptor, with selectivity of 414x for CB2 over CB1,[1] although it is still not as selective as newer agents such as HU-308.
It produces some similar effects to other cannabinoid agonists such as analgesia, but with little or no sedative or psychoactive effects due to its weak CB1 activity, and a relatively strong antiinflammatory effect due to its strong activity at CB2.[2][3]
See also
References
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